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- B4678 CPI-1691 CitationTarget: EZH2|EZH1Summary: EZH2抑制剂
- B1583 UNC19992 CitationTarget: EZH2|EZH1Summary: EZH2抑制剂
- A1615 GANT611 CitationTarget: GLISummary: GLI拮抗剂
- B5859 Entrectinib中文名: 恩曲替尼Target: Trk Receptors|ALK|ROS1Summary: ALK激酶抑制剂
- B4882 PF-06463922中文名: 劳拉替尼Target: ALK|ROS1Summary: ALK/ROS1的强效选择性抑制剂