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- A5573 Pimasertib (AS-703026)Target: MEKSummary: MEK1/2抑制剂
- A8374 AZD8330Target: MEKSummary: MEK 1/2抑制剂
- A8171 Entinostat (MS-275,SNDX-275)2 Citation中文名: 恩替诺特Target: Histone Deacetylases (HDACs)Summary: HDAC1和HDAC3抑制剂
- A3723 Phloretin中文名: 根皮素Target: SGLTSummary: 在苹果中发现的二氢查耳酮
- A4221 YM1552 CitationTarget: SurvivinSummary: Survivin抑制剂,细胞凋亡抑制剂
- A1907 5-Azacytidine6 Citation中文名: 氮胞苷(5-氮胞苷)Target: DNA MethyltransferasesSummary: DNA甲基转移酶抑制剂
- B6342 H-7 dihydrochlorideTarget: PKC|PKG|PKA|Myosin light chain kinases (MLCKs)Summary: 蛋白激酶抑制剂
- A5790 Cidofovir中文名: 西多福韦Target: CMVSummary: 抗CMV药;病毒DNA合成抑制剂
- A4330 Isotretinoin中文名: 罗可坦,异维A酸Target: RARsSummary: 多巴胺β-羟化酶激活剂
- A4064 NVP-BEP800Target: HSP90Summary: 全合成的HSP90β口服抑制剂