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- A8651 LY2940680Target: Smoothened receptorSummary: Hedgehog / SMO拮抗剂,抑制Hh信号。
- A8182 3-Deazaneplanocin A (DZNep) hydrochloride1 Citation中文名: 3-去氮腺嘌呤A盐酸盐Target: EZH2Summary: SAHH和EZH2抑制剂
- A4171 EPZ0056872 CitationTarget: EZH2Summary: EZH2抑制剂
- A4125 CYC116Target: Aurora Kinases|FLT3|VEGFRSummary: Aurora A/B抑制剂
- A3850 TAK-2427 Citation中文名: 瑞沙托维Target: Toll-like receptors (TLRs)|NO Donors / Precursors|IL ReceptorsSummary: TLR 4信号抑制剂
- A3847 SU5416中文名: 司马沙尼Target: VEGFRSummary: VEGF受体抑制剂和AHR激动剂
- A8313 RAF265Target: Raf|VEGFRSummary: 多细胞激酶抑制剂