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- A8651 LY2940680Target: Smoothened receptorSummary: Hedgehog / SMO拮抗剂,抑制Hh信号。
- A8182 3-Deazaneplanocin A (DZNep) hydrochloride1 Citation中文名: 3-去氮腺嘌呤A盐酸盐Target: EZH2Summary: SAHH和EZH2抑制剂
- A4171 EPZ0056872 CitationTarget: EZH2Summary: EZH2抑制剂
- A4170 EPZ004777Target: DOT1LSummary: DOT1L抑制剂
- A8525 Sotrastaurin (AEB071)Target: PKCSummary: PKC抑制剂
- B1287 Ro 31-8220Target: PKCSummary: Pan-PKC抑制剂