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- A4170 EPZ004777Target: DOT1LSummary: DOT1L抑制剂
- A3317 Clozapine N-oxide(CNO)1 Citation中文名: 氯氮平的N-氧化物Target: DREADD LigandsSummary: Clozapine代谢产物,用于化学遗传学
- A4203 Tenovin-1Target: Sir2-like Family Deacetylases (Sirtuins)|p53|p21Summary: SIRT2 抑制剂,p53激活剂
- A1748 Ramelteon1 Citation中文名: 雷美替胺Target: Melatonin ReceptorsSummary: MT1/MT2激动剂