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- A4149 S-Ruxolitinib (INCB018424)中文名: 鲁索替尼Target: JAKSummary: JAK1/2抑制剂
- A8524 Sodium Orthovanadate中文名: 正钒酸钠Target: Protein Tyrosine Phosphatases|alkaline phosphatases|ATPasesSummary: PTP抑制剂
- A8349 Omecamtiv mecarbilTarget: MyosinSummary: 心肌肌球蛋白激活剂
- B1374 WZ4003Target: NUAK1|NUAK2Summary: NUAK1/2抑制剂
- A4140 WP1066Target: STAT|JAKSummary: 细胞通透的JAK2/STAT3抑制剂。