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- A3895 TUG-770Target: Free Fatty Acid ReceptorsSummary: FFA1/GPR40激动剂
- A1709 GW9508Target: Free Fatty Acid ReceptorsSummary: FFA1/GPR40激动剂
- B2014 Probenecid1 Citation中文名: 丙磺舒Target: Organic anion transporters (OATs)|TRP ChannelSummary: 生物学活性
- B7792 AH 76141 CitationTarget: Free Fatty Acid ReceptorsSummary: FFA4/GPR120拮抗剂
- A3145 Afatinib dimaleate中文名: 马来酸阿法替尼Target: EGFR|HER2Summary: EGFR抑制剂
- A8528 TAK-285Target: EGFR|HER2Summary: HER2/EGFR(HER1)抑制剂
- A8366 ARRY-380Target: HER2Summary: 酪氨酸激酶HER2和P95-HER2抑制剂。