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- A8626 ETP-46464Target: PI3K|mTOR|DNA-PK|ATM/ATRSummary: ATR抑制剂
- A1769 KU-00606481 CitationTarget: PI3K|DNA-PKSummary: DNA-PK/PI3-K双重抑制剂
- A8813 NSC697923Target: Ub-conjugating enzyme (E2) complexSummary: E2复合体Ubc13-Uev1A抑制剂
- B2178 BAY 80-6946 (Copanlisib)1 Citation中文名: 库潘尼西Target: PI3KSummary: PI3K抑制剂
- B1572 LatrepirdineTarget: Voltage-gated Calcium Channels (CaV)|NMDA receptor|adrenergic receptor|Histamine receptors|GluR|5-HT receptor|dopamine receptors|AMPA receptorSummary: 脑细胞死亡抑制剂
- A3005 CAL-101 (Idelalisib, GS-1101)2 Citation中文名: 艾代拉里斯,艾代拉利司Target: PI3KSummary: PI3K抑制剂