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- A2412 CP-724714Target: VEGFR|PDGFR|Bcr-Abl|Src|EGFR|c-MET|Insulin Receptors|IRG-1RSummary: 有效的HER2选择性抑制剂
- A4130 ENMD-2076Target: Aurora Kinases|FLT3|RET|Src|VEGFR3/FLT4|NTRK1/TRKA|CSF-1R/c-FmsSummary: Aurora A/Flt3的选择性抑制剂
- A3125 5-Iodotubercidin中文名: 5-碘杀结核菌素Target: Adenosine KinasesSummary: 腺苷激酶抑制剂
- B5298 ABT 702 dihydrochlorideTarget: Adenosine KinasesSummary: 腺苷激酶抑制剂
- B3209 TriapineTarget: Ribonucleotide ReductasesSummary: 核糖核苷酸还原酶(ribonucleotide reductase)抑制剂