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- A8463 Lithocholic Acid中文名: 石胆酸Target: Farnesoid X receptors (FXRs)|Vitamin D receptors (VDRs)|Pregnane X receptor(PXR)Summary: 维生素D受体PXR和FXR的激活剂
- A8215 PP 1Target: Src|EGFR|JAK|ZAP-70Summary: Src家族酪氨酸激酶抑制剂
- A4124 TAK-901Target: Aurora Kinases|FLT3|Src|JAK|LRRK2|Hck|FGR|YES|Fyn|ARGSummary: Aurora A/B抑制剂
- A4511 Cercosporamide中文名: 尾孢素酰胺Target: JAK|MNKSummary: Mnk2和JAK3抑制剂
- A8182 3-Deazaneplanocin A (DZNep) hydrochloride1 Citation中文名: 3-去氮腺嘌呤A盐酸盐Target: EZH2Summary: SAHH和EZH2抑制剂
- A4171 EPZ0056872 CitationTarget: EZH2Summary: EZH2抑制剂
- A4135 Tofacitinib (CP-690550) Citrate2 Citation中文名: 托法替尼Target: JAKSummary: JAK抑制剂
- A4136 TG101348 (SAR302503)2 Citation中文名: 费德拉替尼Target: FLT3|JAK|c-RETSummary: JAK-2抑制剂
- A4137 AZD1480Target: JAKSummary: 新型的ATP竞争性JAK2抑制剂
- A4144 AZ 960Target: JAKSummary: JAKs(janus相关激酶)抑制剂