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- A1185 BMS-754807Target: Insulin and Insulin-like ReceptorsSummary: 有效的、选择性的IGF-1R和InsR抑制剂
- A8440 GSK1838705ATarget: Insulin and Insulin-like Receptors|ALKSummary: ATP竞争性IGF-IR/IR/ALK抑制剂
- A2412 CP-724714Target: VEGFR|PDGFR|Bcr-Abl|Src|EGFR|c-MET|Insulin Receptors|IRG-1RSummary: 有效的HER2选择性抑制剂
- A1302 GSK1904529ATarget: Insulin and Insulin-like ReceptorsSummary: IGF-1R/IR 选择性抑制剂
- A8814 NH1251 CitationTarget: eEF-2Summary: 选择性eEF-2激酶抑制剂
- B1837 Sodium Monofluorophosphate中文名: 单氟磷酸钠Target: phosphatases|Pyruvate kinasesSummary: 丙酮酸激酶和碱性磷酸酶抑制剂
- A3191 Ascomycin(FK 520)中文名: 长川霉素Target: phosphatasesSummary: FK-520 类似物,大环内酯类免疫抑制剂