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- A4333 CPI-6131 CitationTarget: Pyruvate dehydrogenases (PDH)Summary: PDH/α-KGDH抑制剂
- A8313 RAF265Target: Raf|VEGFRSummary: 多细胞激酶抑制剂
- A1832 Doxorubicin (Adriamycin) HCl2 Citation中文名: 盐酸多柔比星,盐酸阿霉素Target: TopoisomerasesSummary: 抗肿瘤抗生素,抑制TOPO II。
- A8412 Dinaciclib (SCH727965)2 CitationTarget: Cyclin-Dependent KinasesSummary: CDK抑制剂
- A5700 BS-181 HClTarget: Cyclin-Dependent KinasesSummary: CDK7抑制剂
- A8252 Nintedanib (BIBF 1120)3 Citation中文名: 尼达尼布Target: VEGFR|PDGFR|FGFRSummary: VEGFR/PDGFR/FGFR抑制剂