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- A4203 Tenovin-1Target: Sir2-like Family Deacetylases (Sirtuins)|p53|p21Summary: SIRT2 抑制剂,p53激活剂
- A8218 Lapatinib2 Citation中文名: 拉帕替尼Target: ErbBSummary: EGFR/HER2抑制剂
- A8375 AZD8931 (Sapitinib)中文名: 沙普替尼Target: EGFR|ErbBSummary: ErbB抑制剂
- A3895 TUG-770Target: Free Fatty Acid ReceptorsSummary: FFA1/GPR40激动剂
- A8506 Potassium CanrenoateTarget: Aldosterone receptorSummary: 醛固酮拮抗剂
- A4092 CUDC-1011 CitationTarget: Histone Deacetylases (HDACs)|EGFR|ErbBSummary: 多靶点HDAC抑制剂
- A4182 Resveratrol2 Citation中文名: 白藜芦醇Target: Sir2-like Family Deacetylases (Sirtuins)|COX|LOX|Adenylyl cyclase|Quinone reductaseSummary: SIRT1激活剂
- B7443 (5Z)-7-Oxozeaenol1 CitationTarget: TAK1Summary: TAK1促分裂原活化蛋白激酶激酶激酶(MAPKKK)抑制剂
- A8319 Dacomitinib (PF299804, PF299)中文名: 达克替尼Target: ErbBSummary: HER抑制剂
- A1709 GW9508Target: Free Fatty Acid ReceptorsSummary: FFA1/GPR40激动剂