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- A3196 AT-101中文名: (R)-(-)-棉子酚Target: NS3/4a ProteasesSummary: BH3-类似物,棉酚对映异构体
- A2678 SU112742 CitationTarget: METSummary: C-Met抑制剂
- A8616 A-674563Target: Cyclin-Dependent Kinases|Akt|GSK-3|ERK|PKC|PKA|RSKSummary: Akt1 / PKA / CDK2的强效选择性抑制剂
- A5703 BMS-777607Target: METSummary: 强效的c-Met选择性抑制剂
- A3573 LY2801653Target: METSummary: MET抑制剂
- A8325 Tivantinib (ARQ 197)2 CitationTarget: METSummary: C-Met抑制剂
- A5354 Zonisamide中文名: 唑尼沙胺Target: Voltage-gated Sodium (NaV) Channels|Voltage-gated Calcium Channels (CaV)|Carbonic Anhydrases|Calcium-Activated Potassium (KCa) ChannelsSummary: 抗惊厥和机械效应的抗癫痫药
- A4364 Methazolamide中文名: 醋甲唑胺Target: Carbonic AnhydrasesSummary: 碳酸酐酶抑制剂
- B1279 Dorzolamide中文名: 多佐胺Target: Carbonic AnhydrasesSummary: 碳酸酐酶抑制剂
- B4904 ACTB-1003Target: VEGFR|FGFR|Tie-2|RSK|p70 S6KSummary: FGFR1抑制剂