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- A4390 Pemetrexed1 Citation中文名: 培美曲塞二钠盐Target: Thymidylate Synthase|DHFR|GARFTSummary: TS、DHFR、GARFT和AICARFT抑制剂
- B6367 NPPBTarget: Calcium-activated chloride channels (CaCC)|GPR35Summary: 氯离子通道抑制剂
- A4069 BMS-707035Target: HIV IntegrasesSummary: HIV-1整合酶抑制剂
- A4070 Elvitegravir (GS-9137)中文名: 埃替格韦Target: HIV IntegrasesSummary: HIV-1整合酶抑制剂
- B4877 URMC-099Target: MLK3Summary: MLK3抑制剂
- B2114 Mitoxantrone HCl中文名: 米托蒽醌Target: Pim|Topoisomerases|USP|HIV IntegrasesSummary: 拓扑异构酶II抑制剂