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- N1336 Chrysin中文名: 柯因,5,7-二羟黄酮Target: Estrogen and Related Receptors|Hypoxia Inducible Factors (HIFs)Summary: 抗炎和抗肿瘤试剂
- A1307 Letrozole中文名: 来曲唑Target: AromatasesSummary: 非甾体类芳香酶抑制剂。
- A5919 AZD7762Target: ChkSummary: ATP竞争性的检查点激酶抑制剂
- B1437 PF-477736Target: ChkSummary: Chk1抑制剂
- A3291 CCT241533Target: ChkSummary: 有效的Chk2抑制剂
- B1236 BML-277Target: ChkSummary: 有效的Chk2选择性抑制剂
- B6004 PX-478 2HClTarget: Hypoxia Inducible Factors (HIFs)Summary: HIF-1α抑制剂
- A8534 Terfenadine中文名: 特非那定Target: Voltage-gated Potassium (KV) Channels|Histamine H1 Receptors|Inward Rectifier Potassium (Kir) ChannelsSummary: 组胺H1受体拮抗剂
- B5880 CCT244747Target: ChkSummary: CHK1抑制剂
- B1198 CisaprideTarget: Voltage-gated Potassium (KV) Channels|5-HT4 ReceptorSummary: 5-HT4受体激动剂