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- A4482 Pifithrin-μ1 CitationTarget: Autophagy|p53|HSP70Summary: p53结合抑制剂,抗凋亡。
- B1850 Teriflunomide中文名: 特立氟胺Target: Dihydroorotate dehydrogenaseSummary: 二氢乳清酸脱氢酶的抑制剂
- A4069 BMS-707035Target: HIV IntegrasesSummary: HIV-1整合酶抑制剂
- B4894 SP2509Target: Histone DemethylasesSummary: 新型LSD1拮抗剂
- B1579 JIB-041 CitationTarget: Histone DemethylasesSummary: Jumonji组蛋白去甲基化酶抑制剂
- A4070 Elvitegravir (GS-9137)中文名: 埃替格韦Target: HIV IntegrasesSummary: HIV-1整合酶抑制剂
- B2114 Mitoxantrone HCl中文名: 米托蒽醌Target: Pim|Topoisomerases|USP|HIV IntegrasesSummary: 拓扑异构酶II抑制剂