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- A4204 JNJ-26854165 (Serdemetan)1 CitationTarget: p53|HDM2 ubiquitin ligaseSummary: P53激活剂,阻断Mdm2-p53相互作用。
- A4379 Lonafarnib中文名: 洛那法尼Target: FPTaseSummary: 高效且具有选择性的法尼基转移酶抑制剂
- A4443 Gliotoxin1 CitationTarget: 20S proteasomal chymotrypsin|Geranylgeranyltransferase I|FarnesyltransferaseSummary: 20S蛋白酶体抑制剂
- A3327 Costunolide中文名: 木香烃内酯Target: FPTase|TelomerasesSummary: BMM分化抑制剂
- A8813 NSC697923Target: Ub-conjugating enzyme (E2) complexSummary: E2复合体Ubc13-Uev1A抑制剂