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- A3278 Nonivamide (Capsaicin Analog)1 Citation中文名: 香草壬酰胺Target: TRP ChannelSummary: TRPV1受体激动剂
- A1174 AMG-517Target: TRP ChannelSummary: TRPV1拮抗剂
- B4899 BLZ9451 CitationTarget: CSF-1RSummary: CSF-1R激酶抑制剂
- B1055 IcilinTarget: TRP ChannelSummary: TRPM8/ hENaCδ激动剂
- A1493 ABT-751 (E7010)1 CitationTarget: Microtubules/TubulinsSummary: 微管聚合抑制剂,抗有丝分裂。
- B5839 SU6656Target: Src|Lyn|YES|FynSummary: Src 酪氨酸激酶抑制剂
- A1655 GW25801 CitationTarget: CSF-1RSummary: CFMS激酶/CSF-1R抑制剂
- A1630 Epothilone B (EPO906, Patupilone)中文名: 埃博霉素B,帕土匹龙Target: Microtubules/TubulinsSummary: 大环内酯物抗癌试剂
- A3022 Pazopanib (GW-786034)中文名: 帕唑帕尼Target: CSF-1R|VEGFR|PDGFR|c-Kit|FGFRSummary: (GW-786034)VEGFR/PDGFR/FGFR 的抑制剂。
- B3270 MMAFTarget: Microtubules/TubulinsSummary: 抗有丝分裂/抗微管蛋白/抗肿瘤剂