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- A1185 BMS-754807Target: Insulin and Insulin-like ReceptorsSummary: 有效的、选择性的IGF-1R和InsR抑制剂
- A8440 GSK1838705ATarget: Insulin and Insulin-like Receptors|ALKSummary: ATP竞争性IGF-IR/IR/ALK抑制剂
- B2223 Zalcitabine中文名: 扎西他滨Target: Reverse TranscriptasesSummary: 逆转录酶抑制剂
- A3608 MK 0893Target: Insulin and Insulin-like Receptors|Glucagon ReceptorsSummary: 胰高血糖素受体/ IGF-1R拮抗剂
- A1755 Tenofovir Disoproxil Fumarate中文名: 富马酸替诺福韦酯Target: Reverse TranscriptasesSummary: 抗逆转录制剂(HIV-1 RT 抑制剂)
- B1946 Foscarnet Sodium中文名: 膦甲酸钠Target: Reverse Transcriptases|RNA PolymerasesSummary: 逆转录酶抑制剂
- B5843 CTX0294885Target: KinasesSummary: Pan-激酶抑制剂
- B2249 Lamotrigine1 Citation中文名: 拉莫三嗪Target: 5-HT receptors|sodium channelSummary: 5-HT抑制剂,钠通道阻断剂
- B2278 Ibutilide Fumarate中文名: 富马酸伊布利特Target: Voltage-gated Potassium (KV) Channels|Voltage-gated Calcium Channels (CaV)|sodium channelSummary: III类抗心律失常药物
- B1789 Mexiletine HCl中文名: 盐酸美西律Target: sodium channelSummary: 钠通道抑制剂