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- A8366 ARRY-380Target: HER2Summary: 酪氨酸激酶HER2和P95-HER2抑制剂。
- B6801 SCH 79797 dihydrochlorideTarget: PARsSummary: PAR1受体拮抗剂
- B5780 UAMC 00039 dihydrochlorideTarget: Dipeptidyl-peptidase IISummary: 二肽基肽酶II(DPP-II)抑制剂
- A3899 UK-50991 CitationTarget: Monocarboxylate transporters (MCTs)|mitochondrial pyruvate carrier (MPC)Summary: MCTs和MPC抑制剂
- A3185 AR-C155858Target: Monocarboxylate transporters (MCTs)Summary: MCT1和MCT2抑制剂
- A3145 Afatinib dimaleate中文名: 马来酸阿法替尼Target: EGFR|HER2Summary: EGFR抑制剂
- A8528 TAK-285Target: EGFR|HER2Summary: HER2/EGFR(HER1)抑制剂