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- A8366 ARRY-380Target: HER2Summary: 酪氨酸激酶HER2和P95-HER2抑制剂。
- B3288 APY29Target: Inositol-requiring enzyme 1 (IRE1)Summary: IRE1α变构调节剂
- B1874 4μ8C2 CitationTarget: Inositol-requiring enzyme 1 (IRE1)Summary: IRE1 Rnase抑制剂
- B3278 BQ-788 sodium salt1 CitationTarget: Endothelin receptorsSummary: ET B受体拮抗剂
- B5624 STF 083010Target: Inositol-requiring enzyme 1 (IRE1)Summary: IRE1α核酸内切酶抑制剂
- A3342 D44761 CitationTarget: CK1Summary: CK1/ALK5抑制剂
- A3719 PF-670462Target: CK1Summary: CK1 ε/δ抑制剂
- A3145 Afatinib dimaleate中文名: 马来酸阿法替尼Target: EGFR|HER2Summary: EGFR抑制剂
- A8528 TAK-285Target: EGFR|HER2Summary: HER2/EGFR(HER1)抑制剂