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- B7072 2-Pyridylethylamine dihydrochlorideTarget: Histamine H1 ReceptorsSummary: 组胺H1受体激动剂
- A8218 Lapatinib2 Citation中文名: 拉帕替尼Target: ErbBSummary: EGFR/HER2抑制剂
- A8375 AZD8931 (Sapitinib)中文名: 沙普替尼Target: EGFR|ErbBSummary: ErbB抑制剂
- A3316 Clemizole hydrochloride中文名: 盐酸克立咪唑Target: Histamine H1 Receptors|TRPC channelSummary: H1组胺受体拮抗剂
- B1566 Rupatadine Fumarate1 Citation中文名: 富马酸卢帕他定Target: Histamine H1 Receptors|PAFRSummary: PAF和组胺(H1)受体的抑制剂
- B4989 EPZ015666Target: Protein Arginine MethyltransferasesSummary: PRMT5抑制剂
- A4092 CUDC-1011 CitationTarget: Histone Deacetylases (HDACs)|EGFR|ErbBSummary: 多靶点HDAC抑制剂
- B3278 BQ-788 sodium salt1 CitationTarget: Endothelin receptorsSummary: ET B受体拮抗剂
- A8319 Dacomitinib (PF299804, PF299)中文名: 达克替尼Target: ErbBSummary: HER抑制剂
- B1568 Azelastine HCl中文名: 盐酸氮卓斯汀Target: Histamine H1 ReceptorsSummary: 有效的,第二代,选择性的组胺受体拮抗剂