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- A3237 Betulinic acid中文名: 白桦脂酸,桦木酸Target: Aminopeptidases|Topoisomerases|HIVSummary: 抗HIV和抗肿瘤化合物,五环三萜类化合物
- B2157 Cabazitaxel3 Citation中文名: 卡巴他赛Target: Microtubule/TubulinSummary: 微管相关抑制剂
- A1765 Vincristine sulfate中文名: 硫酸长春新碱Target: Microtubule/TubulinSummary: 微管的破坏者,抗肿瘤剂
- B4745 (S)-10-Hydroxycamptothecin中文名: 羟喜树碱Target: TopoisomerasesSummary: 拓扑异构酶I抑制剂
- B5743 SR 2211Target: Retinoic acid-related Orphan Receptors (RORs)Summary: RORγ反向激动剂
- A3394 Epothilone D中文名: 埃博霉素 DTarget: Microtubule/TubulinSummary: 天然聚酮化合物
- B1463 KPT-276Target: nuclear export|CRM1Summary: CRM1抑制剂
- A8400 Clinafloxacin CI96 AM1091中文名: 克林沙星Target: TopoisomerasesSummary: 拓扑异构酶抑制剂
- A2601 Aclacinomycin ATarget: TopoisomerasesSummary: 拓扑异构酶I和II的双重抑制剂
- N2133 7-Ethyl-10-hydroxycamptothecinTarget: TopoisomerasesSummary: TOPO I抑制剂