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- A3237 Betulinic acid中文名: 白桦脂酸,桦木酸Target: Aminopeptidases|Topoisomerases|HIVSummary: 抗HIV和抗肿瘤化合物,五环三萜类化合物
- B4745 (S)-10-Hydroxycamptothecin中文名: 羟喜树碱Target: TopoisomerasesSummary: 拓扑异构酶I抑制剂
- B5743 SR 2211Target: Retinoic acid-related Orphan Receptors (RORs)Summary: RORγ反向激动剂
- B1463 KPT-276Target: nuclear export|CRM1Summary: CRM1抑制剂
- A5588 Oligomycin A1 Citation中文名: 寡霉素ATarget: Synthases/SynthetasesSummary: 线粒体ATP合成酶抑制剂
- B1472 Mizoribine中文名: 咪唑立宾Target: Synthases/SynthetasesSummary: DNA/RNA合成抑制剂
- A2402 Floxuridine中文名: 氟尿苷Target: Synthases/SynthetasesSummary: 抗肿瘤抗代谢物
- B7070 Triacsin CTarget: Synthases/SynthetasesSummary: 酰基辅酶A合成酶抑制剂
- A8432 Fenticonazole Nitrate中文名: 硝酸芬替康唑Target: Cytochrome P450 (CYP450)|Synthases/SynthetasesSummary: 抗真菌药
- A8400 Clinafloxacin CI96 AM1091中文名: 克林沙星Target: TopoisomerasesSummary: 拓扑异构酶抑制剂