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- N1336 Chrysin中文名: 柯因,5,7-二羟黄酮Target: Estrogen and Related Receptors|Hypoxia Inducible Factors (HIFs)Summary: 抗炎和抗肿瘤试剂
- A3358 DeltarasinTarget: Phosphodiesterases (PDEs)Summary: KRAS-PDEδ相互作用抑制剂
- B1386 Milrinone中文名: 米力农Target: Phosphodiesterases (PDEs)Summary: PDE3抑制剂
- B6004 PX-478 2HClTarget: Hypoxia Inducible Factors (HIFs)Summary: HIF-1α抑制剂
- B7157 OGT 2115Target: HeparanasesSummary: 乙酰肝素酶抑制剂
- B1471 Adenine HCl中文名: 腺嘌呤盐酸盐Target: Adenine receptorsSummary: 腺苷受体激动剂
- B1115 BAY 87-2243Target: Hypoxia Inducible Factors (HIFs)Summary: 有效的HIF-1选择性抑制剂
- A4346 Aminophylline中文名: 氨茶碱,氨基非林Target: Phosphodiesterases (PDEs)Summary: Pan-PDE抑制剂
- A4334 Avanafil中文名: 阿伐那非Target: Phosphodiesterases (PDEs)Summary: PDE5抑制剂
- A4325 PF-2545920Target: Phosphodiesterases (PDEs)Summary: PDE10A的有效选择性抑制剂