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- N1336 Chrysin中文名: 柯因,5,7-二羟黄酮Target: Estrogen and Related Receptors|Hypoxia Inducible Factors (HIFs)Summary: 抗炎和抗肿瘤试剂
- A4356 Varespladib (LY315920)中文名: 伐瑞拉迪Target: PhospholipasesSummary: HnsPLA的强效选择性抑制剂
- A1493 ABT-751 (E7010)1 CitationTarget: Microtubules/TubulinsSummary: 微管聚合抑制剂,抗有丝分裂。
- A4491 SGC-CBP302 CitationTarget: CREBBP|EP300Summary: CREBBP/EP300 bromodomain抑制剂
- A1630 Epothilone B (EPO906, Patupilone)中文名: 埃博霉素B,帕土匹龙Target: Microtubules/TubulinsSummary: 大环内酯物抗癌试剂
- B6004 PX-478 2HClTarget: Hypoxia Inducible Factors (HIFs)Summary: HIF-1α抑制剂
- B3270 MMAFTarget: Microtubules/TubulinsSummary: 抗有丝分裂/抗微管蛋白/抗肿瘤剂
- A4490 I-CBP 112Target: CREBBP|EP300Summary: CBP/EP300 bromodomain抑制剂
- B1823 Quinacrine 2HCl中文名: 盐酸奎纳克林Target: Phospholipases|Monoamine oxidases (MAOs)Summary: 抗原虫剂
- B1115 BAY 87-2243Target: Hypoxia Inducible Factors (HIFs)Summary: 有效的HIF-1选择性抑制剂