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- A3237 Betulinic acid中文名: 白桦脂酸,桦木酸Target: Aminopeptidases|Topoisomerases|HIVSummary: 抗HIV和抗肿瘤化合物,五环三萜类化合物
- A2575 Bestatin中文名: 乌苯美司Target: AminopeptidasesSummary: 氨肽酶抑制剂
- A4355 Tosedostat (CHR2797)1 Citation中文名: 托舍多特Target: AminopeptidasesSummary: 氨肽酶(Aminopeptidase)抑制剂
- A2917 Flumazenil中文名: 氟马西尼Target: GABAA ReceptorsSummary: 苯二氮卓拮抗剂
- B4745 (S)-10-Hydroxycamptothecin中文名: 羟喜树碱Target: TopoisomerasesSummary: 拓扑异构酶I抑制剂
- B8015 ML216Target: BLMSummary: BLM解旋酶抑制剂
- A8435 Furosemide中文名: 呋塞米Target: Na /K /Cl- Symporters (NKCCs)|GABAA ReceptorsSummary: GABAA受体拮抗剂
- N1592 (+)-Bicuculline中文名: 荷包牡丹碱Target: GABAA Receptors|Calcium-Activated Potassium (KCa) ChannelsSummary: GABAA受体拮抗剂
- A8400 Clinafloxacin CI96 AM1091中文名: 克林沙星Target: TopoisomerasesSummary: 拓扑异构酶抑制剂
- A2601 Aclacinomycin ATarget: TopoisomerasesSummary: 拓扑异构酶I和II的双重抑制剂