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- A8366 ARRY-380Target: HER2Summary: 酪氨酸激酶HER2和P95-HER2抑制剂。
- B6367 NPPBTarget: Calcium-activated chloride channels (CaCC)|GPR35Summary: 氯离子通道抑制剂
- B5410 AZ 10606120 dihydrochlorideTarget: P2X ReceptorsSummary: P2X7受体拮抗剂
- A3136 A-740003Target: P2X ReceptorsSummary: P2X7受体拮抗剂
- A8180 KN-62Target: Ca2 /calmodulin-dependent protein kinases (CaMKs)|P2X ReceptorsSummary: 钙调蛋白激酶II抑制剂
- A3145 Afatinib dimaleate中文名: 马来酸阿法替尼Target: EGFR|HER2Summary: EGFR抑制剂
- A8528 TAK-285Target: EGFR|HER2Summary: HER2/EGFR(HER1)抑制剂