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- A2571 Pepstatin A1 Citation中文名: 抑肽素Target: Cathepsins|Renin|HIV proteases|PepsinsSummary: 天冬氨酸蛋白酶抑制剂
- B2014 Probenecid1 Citation中文名: 丙磺舒Target: Organic anion transporters (OATs)|TRP ChannelSummary: 生物学活性
- B1055 IcilinTarget: TRP ChannelSummary: TRPM8/ hENaCδ激动剂
- A3278 Nonivamide (Capsaicin Analog)1 Citation中文名: 香草壬酰胺Target: TRP ChannelSummary: TRPV1受体激动剂
- A1174 AMG-517Target: TRP ChannelSummary: TRPV1拮抗剂
- A8189 PSI-62063 CitationTarget: HCV polymeraseSummary: HCV RNA聚合酶抑制剂
- A3738 PSI-7977中文名: 索非布韦,索氟布韦Target: HCV polymeraseSummary: 慢性丙型肝炎病毒(HCV)感染的抗病毒剂
- A4032 VX-222 (VCH-222, Lomibuvir)Target: HCV polymeraseSummary: HCV RNA聚合酶抑制剂