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- A3021 GDC-0449 (Vismodegib)1 Citation中文名: 维莫德吉Target: P-glycoprotein (P-gp)|HedgehogSummary: Hedgehog拮抗剂
- A8245 Sorafenib Tosylate1 Citation中文名: 甲苯磺酸索拉非尼Target: Raf|VEGFRSummary: Raf激酶和酪氨酸激酶抑制剂
- B1174 LGX818中文名: 康奈非尼Target: RafSummary: RAF抑制剂
- A3196 AT-101中文名: (R)-(-)-棉子酚Target: NS3/4a ProteasesSummary: BH3-类似物,棉酚对映异构体
- A8313 RAF265Target: Raf|VEGFRSummary: 多细胞激酶抑制剂