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- B4572 β-Estradiol - d3Target: Estrogen and Related ReceptorsSummary: 氘代β雌二醇
- A2412 CP-724714Target: VEGFR|PDGFR|Bcr-Abl|Src|EGFR|c-MET|Insulin Receptors|IRG-1RSummary: 有效的HER2选择性抑制剂
- B1394 Tamoxifen Citrate中文名: 枸橼酸他莫昔Target: Estrogen and Related ReceptorsSummary: 抗雌激素药
- B1507 Estriol中文名: 雌三醇Target: Estrogen and Related ReceptorsSummary: 雌激素受体拮抗剂
- A3173 AMD-070Target: CXCRSummary: CXCR4拮抗剂
- B3266 AMG 4871 CitationTarget: CXCRSummary: CXCR3拮抗剂
- A3753 Reparixin L-lysine salt1 Citation中文名: 瑞帕利辛L-赖氨酸盐Target: CXCRSummary: CXCL8受体CXCR1/CXCR2活化的抑制剂
- A3803 SCH 563705Target: CXCRSummary: CXCR2/CXCR1拮抗剂
- B1506 Estradiol valerate中文名: 戊酸雌二醇Target: Estrogen and Related ReceptorsSummary: 雌激素受体激动剂
- B1513 Toremifene Citrate中文名: 枸橼酸托瑞米芬Target: Estrogen and Related ReceptorsSummary: 口服选择性雌激素受体调节剂(SERM)