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- A3965 BI 25361 CitationTarget: PLK|Bromodomain-containing proteins(BRDs)Summary: ATP竞争性的Plk1抑制剂
- A1905 3-Deazaneplanocin,DZNep6 Citation中文名: 3-去氮腺嘌呤ATarget: HydrolaseSummary: S-腺苷高半胱氨酸和EZH2抑制剂。
- B1288 RigosertibTarget: PI3K|PLKSummary: PI3K/PLK1抑制剂
- A8681 Ro3280Target: PLKSummary: PLK1高选择性抑制剂
- B7661 DLPCTarget: Nuclear ReceptorsSummary: LRH-1激动剂配体