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- A3012 Ruxolitinib (INCB018424)4 Citation中文名: 鲁索替尼Target: JAKSummary: JAK抑制剂
- A4090 JNJ-264815853 CitationTarget: Histone Deacetylases (HDACs)Summary: HDAC抑制剂
- A8171 Entinostat (MS-275,SNDX-275)2 Citation中文名: 恩替诺特Target: Histone Deacetylases (HDACs)Summary: HDAC1和HDAC3抑制剂
- A4112 Barasertib (AZD1152-HQPA)3 Citation中文名: 巴拉塞替Target: Aurora KinasesSummary: Aurora Kinase B抑制剂
- A8214 AZD80552 CitationTarget: mTORSummary: MTOR 抑制剂
- B2127 Rifapentine中文名: 利福喷丁Target: RNA PolymerasesSummary: 治疗肺结核的抗生素药物.
- A3021 GDC-0449 (Vismodegib)1 Citation中文名: 维莫德吉Target: P-glycoprotein (P-gp)|HedgehogSummary: Hedgehog拮抗剂
- A8346 BYL-7191 Citation中文名: 阿培利司Target: PI3KSummary: 选择性的PI3Kα抑制剂
- N2791 Cucurbitacin E中文名: 葫芦素 ETarget: ActinSummary: 抑制肌动蛋白解聚
- B7070 Triacsin CTarget: Synthases/SynthetasesSummary: 酰基辅酶A合成酶抑制剂