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- A4010 Salinosporamide A (NPI-0052, Marizomib)Target: ProteasomeSummary: 20S蛋白酶体抑制剂
- A8163 AM 1142 CitationTarget: ProteasomeSummary: 20S蛋白酶体抑制剂
- A4011 ONX-0914 (PR-957)6 CitationTarget: ProteasomeSummary: 免疫蛋白酶体(immunoproteasome)抑制剂
- A3253 BMS-6265292 CitationTarget: HIV-1 gp120Summary: HIV-1吸附的抑制剂
- A1909 BIX 01294Target: G9aSummary: G9a和GLP抑制剂
- B6026 VR23Target: ProteasomeSummary: 蛋白酶抑制剂
- A2578 Clasto-Lactacystin β-lactoneTarget: ProteasomeSummary: 蛋白酶体抑制剂
- B1492 PYR-412 CitationTarget: ProteasomeSummary: 泛素活化酶(E1)抑制剂
- B7757 UNC 0642Target: G9a|GLPSummary: G9a和GLP组蛋白赖氨酸甲基转移酶抑制剂
- A2604 Celastrol中文名: 雷公藤红素Target: ProteasomeSummary: 抗氧化、抗炎和免疫抑制剂