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- B1135 GDC-0623Target: MEKSummary: MEK1抑制剂
- A4203 Tenovin-1Target: Sir2-like Family Deacetylases (Sirtuins)|p53|p21Summary: SIRT2 抑制剂,p53激活剂
- A4325 PF-2545920Target: Phosphodiesterases (PDEs)Summary: PDE10A的有效选择性抑制剂
- A8340 Cyclopamine1 Citation中文名: 环巴胺Target: SmoothenedSummary: Hedgehog (Hh)信号抑制剂