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- A3962 AZD1208Target: PimSummary: PIM激酶抑制剂
- A4390 Pemetrexed1 Citation中文名: 培美曲塞二钠盐Target: Thymidylate Synthase|DHFR|GARFTSummary: TS、DHFR、GARFT和AICARFT抑制剂
- A8178 Panobinostat (LBH589)10 Citation中文名: 帕比司他Target: Histone Deacetylases (HDACs)Summary: HDAC抑制剂
- A4325 PF-2545920Target: Phosphodiesterases (PDEs)Summary: PDE10A的有效选择性抑制剂
- A8183 Trichostatin A (TSA)13 Citation中文名: 曲古柳菌素ATarget: Histone Deacetylases (HDACs)Summary: HDAC抑制剂
- A4098 PCI-24781 (CRA-024781)Target: Histone Deacetylases (HDACs)Summary: Pan-HDAC抑制剂