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- A8637 IOWH-032Target: CFTRSummary: CFTR抑制剂
- A4325 PF-2545920Target: Phosphodiesterases (PDEs)Summary: PDE10A的有效选择性抑制剂
- A8623 TOK-001中文名: 加来特龙,伽来特隆Target: Androgen Receptors|Cytochrome P450 (CYP450)Summary: CYP17抑制剂和雄激素受体(AR)拮抗剂
- A5979 Tie2 kinase inhibitor中文名: Tie2激酶抑制剂Target: Tie-2Summary: Tie-2(Tie2 )抑制剂