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- B6036 INCB-024360中文名: 艾卡哚司他Target: IDOSummary: 强效的IDO1抑制剂
- A1185 BMS-754807Target: Insulin and Insulin-like ReceptorsSummary: 有效的、选择性的IGF-1R和InsR抑制剂
- A5700 BS-181 HClTarget: Cyclin-Dependent KinasesSummary: CDK7抑制剂
- A4203 Tenovin-1Target: Sir2-like Family Deacetylases (Sirtuins)|p53|p21Summary: SIRT2 抑制剂,p53激活剂