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- N2133 7-Ethyl-10-hydroxycamptothecinTarget: TopoisomerasesSummary: TOPO I抑制剂
- A3444 GS-9620中文名: 维沙莫德Target: Toll-like receptors (TLRs)Summary: TLR-7激动剂
- A5161 Imiquimod中文名: 咪喹莫特Target: Toll-like receptors (TLRs)Summary: TLR-7激动剂,具有抗病毒和抗肿瘤活性的免疫调节剂
- A2601 Aclacinomycin ATarget: TopoisomerasesSummary: 拓扑异构酶I和II的双重抑制剂
- B5881 RI-2Target: RAD51Summary: RAD51抑制剂
- B4745 (S)-10-Hydroxycamptothecin中文名: 羟喜树碱Target: TopoisomerasesSummary: 拓扑异构酶I抑制剂
- B1801 Norfloxacin中文名: 诺氟沙星Target: TopoisomerasesSummary: 拓扑异构酶抑制剂
- A4536 Fostriecin sodium saltTarget: PP1|PP2A|Topoisomerases|PP4Summary: 抗肿瘤抗生素
- A8721 CBR-58841 CitationTarget: 3-phosphoglycerate dehydrogenaseSummary: PHGDH抑制剂
- A1832 Doxorubicin (Adriamycin) HCl2 Citation中文名: 盐酸多柔比星,盐酸阿霉素Target: TopoisomerasesSummary: 抗肿瘤抗生素,抑制TOPO II。