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- N2133 7-Ethyl-10-hydroxycamptothecinTarget: TopoisomerasesSummary: TOPO I抑制剂
- B6342 H-7 dihydrochlorideTarget: PKC|PKG|PKA|Myosin light chain kinases (MLCKs)Summary: 蛋白激酶抑制剂
- B6062 Manumycin A中文名: 手霉素ASummary: 法尼基转移酶抑制剂
- A4447 2,3-DCPE hydrochlorideTarget: Apoptosis InducersSummary: Bcl-XL蛋白表达下调剂
- A3023 P0050911 CitationTarget: Ubiquitin-specific proteasesSummary: 泛素特异性蛋白酶7(USP7)抑制剂
- A3785 Salinomycin中文名: 盐霉素(来自白色链霉菌)Target: AntibioticSummary: 聚醚离子载体抗生素,抗癌
- A8236 Regorafenib4 Citation中文名: 瑞戈非尼Target: Raf|VEGFR|PDGFR|c-Kit|RETSummary: VEGFR/PDGFR/FGFR/mutant Kit/RET/Raf-1抑制剂
- A1980 SNS-032 (BMS-387032)2 CitationTarget: Cyclin-Dependent KinasesSummary: CDK抑制剂
- A3016 PLX-47201 CitationTarget: RafSummary: BRAF激酶抑制剂
- B6026 VR23Target: ProteasomeSummary: 蛋白酶抑制剂