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Signaling Pathways - DREADD Ligands - NTRK1/TRKA - Nrf2/ARE signal - Carbonic Anhydrases

10 件产品

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  1. Dorzolamide
    B1279 Dorzolamide
    中文名: 多佐胺
    Target: Carbonic Anhydrases
    Summary: 碳酸酐酶抑制剂
      Soluble in DMSO
  2. Chlorothiazide
    A8397 Chlorothiazide
    中文名: 氯噻嗪
    Target: Carbonic Anhydrases
    Summary: 碳酸酐酶抑制剂
      ≥14.85 mg/mL
      insoluble in H2O
  3. Methyocarbamol
    A8473 Methyocarbamol
    中文名: 美索巴莫
    Target: Carbonic Anhydrases
    Summary: 碳酸酐酶抑制剂
      ≥15.65 mg/mL
      ≥7.7 mg/mL
  4. Zonisamide
    A5354 Zonisamide
    中文名: 唑尼沙胺
    Target: Voltage-gated Sodium (NaV) Channels|Voltage-gated Calcium Channels (CaV)|Carbonic Anhydrases|Calcium-Activated Potassium (KCa) Channels
    Summary: 抗惊厥和机械效应的抗癫痫药
      ≥8.35 mg/mL
      insoluble in H2O
  5. Clozapine N-oxide(CNO)
    A3317 Clozapine N-oxide(CNO)
     1 Citation
    中文名: 氯氮平的N-氧化物
    Target: DREADD Ligands
    Summary: Clozapine代谢产物,用于化学遗传学
      ≥17.15 mg/mL
      ≥49 mg/mL
  6. Methazolamide
    A4364 Methazolamide
    中文名: 醋甲唑胺
    Target: Carbonic Anhydrases
    Summary: 碳酸酐酶抑制剂
      ≥23.63 mg/mL
      ≥2.58 mg/mL
  7. Tioxolone
    A4362 Tioxolone
    中文名: 噻克索酮
    Target: Carbonic Anhydrases
    Summary: CAI抑制剂
      ≥63.2 mg/mL
      ≥2.33 mg/mL
  8. U-104
    A4358 U-104
    Target: Carbonic Anhydrases
    Summary: CAIX抑制剂
      ≥11.5 mg/mL
      insoluble in H2O
  9. ENMD-2076
    A4130 ENMD-2076
    Target: Aurora Kinases|FLT3|RET|Src|VEGFR3/FLT4|NTRK1/TRKA|CSF-1R/c-Fms
    Summary: Aurora A/Flt3的选择性抑制剂
      ≥18.75 mg/mL
      insoluble in H2O
  10. 5,7-dihydroxychromone
    N2172 5,7-dihydroxychromone
     1 Citation
    中文名: 5,7-二羟基色酮
    Target: Nrf2/ARE signal|PPAR
    Summary: Nrf2/ARE信号激活剂和PPARγ激动剂
      ≥7.05 mg/mL
      insoluble in H2O

10 件产品

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