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Signaling Pathways - DREADD Ligands - O6-methylguanine-DNA-methyl-transferase (MGMT) - Glucocorticoid Receptors - PKG

10 件产品

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  1. Methylprednisolone Sodium Succinate
    B4953 Methylprednisolone Sodium Succinate
    中文名: 甲泼尼龙琥珀酸钠
    Target: Glucocorticoid Receptors
    Summary: 糖皮质激素
      ≥49.7 mg/mL
      ≥2.94 mg/mL
  2. H-7 dihydrochloride
    B6342 H-7 dihydrochloride
    Target: PKC|PKG|PKA|Myosin light chain kinases (MLCKs)
    Summary: 蛋白激酶抑制剂
      Soluble in DMSO
  3. Fasudil
    B3523 Fasudil
    中文名: 法舒地尔
    Target: ROCK|PKC|PKG|PKA|Myosin light chain kinases (MLCKs)
    Summary: 钙拮抗剂
      Soluble in DMSO
  4. Fluticasone propionate
    B2096 Fluticasone propionate
    中文名: 丙酸氟替卡松
    Target: Glucocorticoid Receptors
    Summary: 高亲和力,选择性糖皮质激素受体激动剂
      ≥18.5 mg/mL
      insoluble in H2O
  5. Dexamethasone acetate
    B1926 Dexamethasone acetate
    中文名: 醋酸地塞米松
    Target: Glucocorticoid Receptors|interleukin receptor
    Summary: IL受体调节剂
      ≥13.35 mg/mL
      insoluble in H2O
  6. Mifepristone
    B1511 Mifepristone
     3 Citation
    中文名: 美服培酮
    Target: Progesterone Receptors|Glucocorticoid Receptors
    Summary: 孕激素受体拮抗剂
      ≥21.48 mg/mL
      insoluble in H2O
  7. GSK690693
    A5072 GSK690693
    Target: Akt|PKC|PKG|PKA|Prk
    Summary: ATP竞争性的Pan-AKT抑制剂
      ≥21.25 mg/mL
      insoluble in H2O
  8. Clozapine N-oxide(CNO)
    A3317 Clozapine N-oxide(CNO)
     1 Citation
    中文名: 氯氮平的N-氧化物
    Target: DREADD Ligands
    Summary: Clozapine代谢产物,用于化学遗传学
      ≥17.15 mg/mL
      ≥49 mg/mL
  9. Lomeguatrib
    A1912 Lomeguatrib
    中文名: 罗米鲁曲
    Target: O6-methylguanine-DNA-methyl-transferase (MGMT)
    Summary: MGMT抑制剂
      ≥50 mg/mL
      insoluble in H2O
  10. Methylprednisolone
    A4233 Methylprednisolone
    中文名: 甲泼尼龙
    Target: Glucocorticoid Receptors
    Summary: 细胞凋亡诱导剂,GR激动剂
      ≥15.35 mg/mL
      insoluble in H2O

10 件产品

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