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Signaling Pathways - MAGL - TAK1 - sodium channel - Deubiquitinating enzymes (DUBs)

10 件产品

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  1. Spautin-1
    B5873 Spautin-1
     1 Citation
    Target: Deubiquitinating enzymes (DUBs)|Autophagy
    Summary: 自噬抑制剂
      ≥13.5 mg/mL
      insoluble in H2O
  2. (5Z)-7-Oxozeaenol
    B7443 (5Z)-7-Oxozeaenol
     1 Citation
    Target: TAK1
    Summary: TAK1促分裂原活化蛋白激酶激酶激酶(MAPKKK)抑制剂
      <9.06 mg/mL
      insoluble in ethanol
  3. Ibutilide Fumarate
    B2278 Ibutilide Fumarate
    中文名: 富马酸伊布利特
    Target: Voltage-gated Potassium (KV) Channels|Voltage-gated Calcium Channels (CaV)|sodium channel
    Summary: III类抗心律失常药物
      ≥25.6 mg/mL
      ≥16.4 mg/mL
  4. Lamotrigine
    B2249 Lamotrigine
     1 Citation
    中文名: 拉莫三嗪
    Target: 5-HT receptors|sodium channel
    Summary: 5-HT抑制剂,钠通道阻断剂
      ≥12.3 mg/mL
      insoluble in H2O
  5. ML-323
    B1317 ML-323
    Target: Deubiquitinating enzymes (DUBs)
    Summary: USP1-UAF1抑制剂
      ≥15.05 mg/mL
      ≥2.25 mg/mL
  6. PR-619
    A8212 PR-619
    Target: Deubiquitinating enzymes (DUBs)
    Summary: 去泛素化酶(DUBs)抑制剂
      ≥11.15 mg/mL
      insoluble in H2O
  7. NSC 687852 (b-AP15)
    A4453 NSC 687852 (b-AP15)
    Target: Deubiquitinating enzymes (DUBs)
    Summary: 19S调节颗粒抑制剂
      ≥20.95 mg/mL
      insoluble in H2O
  8. Vialinin A
    A4429 Vialinin A
    Target: Deubiquitinating enzymes (DUBs)|IL Receptors|CCL2
    Summary: USP/IsoT/UCH-L1 DUB抑制剂
      Soluble in DMSO
  9. Dronedarone
    A3374 Dronedarone
    中文名: 决奈达隆
    Target: Cytochrome P450 (CYP450)|sodium channel|adrenergic receptor|potassium channel|calcium channel
    Summary: CYP3A4和2D6抑制剂
      ≥27.84 mg/mL
      insoluble in H2O
  10. Tanshinone IIA
    N1846 Tanshinone IIA
    中文名: 丹参酮IIA
    Target: AP-1|MAGL
    Summary: 抗氧化和抗炎剂
      ≥3.42 mg/mL
      insoluble in H2O

10 件产品

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