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Signaling Pathways - Prostaglandin EP receptors - Calpains - Quinone reductase - sodium channel

10 件产品

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  1. Prostaglandin E2
    B7005 Prostaglandin E2
    中文名: 前列腺素E2
    Target: Prostaglandin EP receptors
    Summary: 内源性前列腺素
      ≥42.8 mg/mL
      insoluble in H2O
  2. Ibutilide Fumarate
    B2278 Ibutilide Fumarate
    中文名: 富马酸伊布利特
    Target: Voltage-gated Potassium (KV) Channels|Voltage-gated Calcium Channels (CaV)|sodium channel
    Summary: III类抗心律失常药物
      ≥25.6 mg/mL
      ≥16.4 mg/mL
  3. Lamotrigine
    B2249 Lamotrigine
     1 Citation
    中文名: 拉莫三嗪
    Target: 5-HT receptors|sodium channel
    Summary: 5-HT抑制剂,钠通道阻断剂
      ≥12.3 mg/mL
      insoluble in H2O
  4. PD 150606
    A4413 PD 150606
    Target: Calpains
    Summary: 非肽类钙蛋白酶抑制剂
      Soluble in DMSO
  5. MDL 28170
    A4412 MDL 28170
    Target: Cathepsins|Calpains
    Summary: Calpain和cathepsin B抑制剂
      ≥16.75 mg/mL
      insoluble in H2O
  6. Dronedarone
    A3374 Dronedarone
    中文名: 决奈达隆
    Target: Cytochrome P450 (CYP450)|sodium channel|adrenergic receptor|potassium channel|calcium channel
    Summary: CYP3A4和2D6抑制剂
      ≥27.84 mg/mL
      insoluble in H2O
  7. Resveratrol
    A4182 Resveratrol
     2 Citation
    中文名: 白藜芦醇
    Target: Sir2-like Family Deacetylases (Sirtuins)|COX|LOX|Adenylyl cyclase|Quinone reductase
    Summary: SIRT1激活剂
      ≥9.65 mg/mL
      insoluble in H2O
  8. Calpain Inhibitor I, ALLN
    A2602 Calpain Inhibitor I, ALLN
     2 Citation
    Target: Cathepsins|Calpains
    Summary: Calpain I/II/ B/L抑制剂
      ≥19.1 mg/mL
      insoluble in H2O
  9. E-64
    A2576 E-64
     2 Citation
    Target: Cathepsins|Calpains|Papains
    Summary: 半胱氨酸蛋白酶(cysteine protease)抑制剂
      ≥53.6 mg/mL
      ≥49.1 mg/mL
  10. Leupeptin, Microbial
    A2570 Leupeptin, Microbial
    中文名: 亮抑酶肽
    Target: Cathepsins|Calpains|Trypsins
    Summary: 丝氨酸和半胱氨酸蛋白酶抑制剂
      ≥24.7 mg/mL
      ≥54.4 mg/mL

10 件产品

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