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Signaling Pathways - DGAT - sodium channel - NUAK1 - Thymidylate Synthase

10 件产品

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  1. WZ4003
    B1374 WZ4003
    Target: NUAK1|NUAK2
    Summary: NUAK1/2抑制剂
      ≥7.85 mg/mL
      insoluble in H2O
  2. Raltitrexed
    B1476 Raltitrexed
    中文名: 雷替曲塞
    Target: Thymidylate Synthase
    Summary: 胸苷酸合酶抑制剂
      ≥154 mg/mL
      insoluble in H2O
  3. Ibutilide Fumarate
    B2278 Ibutilide Fumarate
    中文名: 富马酸伊布利特
    Target: Voltage-gated Potassium (KV) Channels|Voltage-gated Calcium Channels (CaV)|sodium channel
    Summary: III类抗心律失常药物
      ≥25.6 mg/mL
      ≥16.4 mg/mL
  4. Lamotrigine
    B2249 Lamotrigine
     1 Citation
    中文名: 拉莫三嗪
    Target: 5-HT receptors|sodium channel
    Summary: 5-HT抑制剂,钠通道阻断剂
      ≥12.3 mg/mL
      insoluble in H2O
  5. MRT67307 HCl
    A3635 MRT67307 HCl
    Target: TBK1|MARK1|NUAK1
    Summary: SIK/TBK-1/IKKe抑制剂
      ≥23.25 mg/mL
      ≥52.5 mg/mL
  6. Dronedarone
    A3374 Dronedarone
    中文名: 决奈达隆
    Target: Cytochrome P450 (CYP450)|sodium channel|adrenergic receptor|potassium channel|calcium channel
    Summary: CYP3A4和2D6抑制剂
      ≥27.84 mg/mL
      insoluble in H2O
  7. AZD7687
    A3215 AZD7687
    Target: DGAT
    Summary: 强效的选择性DGAT抑制剂
      Soluble in DMSO
  8. Pemetrexed
    A4390 Pemetrexed
     1 Citation
    中文名: 培美曲塞二钠盐
    Target: Thymidylate Synthase|DHFR|GARFT
    Summary: TS、DHFR、GARFT和AICARFT抑制剂
      ≥15.68 mg/mL
      ≥30.67 mg/mL
  9. A922500
    A4382 A922500
    Target: DGAT
    Summary: DGAT-1抑制剂
      ≥21.25 mg/mL
      insoluble in H2O
  10. Fluorouracil (Adrucil)
    A4071 Fluorouracil (Adrucil)
     3 Citation
    中文名: 氟尿嘧啶
    Target: Thymidylate Synthase
    Summary: 胸苷酸合成酶抑制剂,抗肿瘤药物。
      ≥13.04 mg/mL
      ≥10.04 mg/mL

10 件产品

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