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Signaling Pathways - Hedgehog - adrenergic receptor - Survivin - MK2

10 件产品

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  1. MK2 Inhibitor IV
    C5545 MK2 Inhibitor IV
    Target: MK2
    Summary: 高选择性、非ATP竞争性MK2抑制剂
      insoluble in DMSO
      ≥37.4 mg/mL
  2. CMPD-1
    B6962 CMPD-1
    Target: Microtubules/Tubulins|MK2
    Summary: p38α介导的MK2a磷酸化的抑制剂
      <34.94 mg/mL
      <34.94 mg/mL
  3. PF-3644022
    B5549 PF-3644022
    Target: MK2
    Summary: MK2抑制剂
      <14.98 mg/mL
  4. Epinephrine Bitartrate
    B1358 Epinephrine Bitartrate
    中文名: 酒石酸肾上腺素
    Target: adrenergic receptor
    Summary: 肾上腺素能受体激动剂
      ≥16.66 mg/mL
      ≥22.9 mg/mL
  5. Latrepirdine
    B1572 Latrepirdine
    Target: Voltage-gated Calcium Channels (CaV)|NMDA receptor|adrenergic receptor|Histamine receptors|GluR|5-HT receptor|dopamine receptors|AMPA receptor
    Summary: 脑细胞死亡抑制剂
      ≥19.62 mg/mL
      insoluble in H2O
  6. Quetiapine
    A3744 Quetiapine
    中文名: 喹硫平
    Target: AChR|adrenergic receptor|5-HT receptor|Dopamine receptor|Histamine receptor
    Summary: 多巴胺受体拮抗剂
      ≥19.18 mg/mL
      insoluble in H2O
  7. PHA-767491
    A3721 PHA-767491
    Target: Cyclin-Dependent Kinases|MK2|Cdc7
    Summary: Cdc7 / CDK9抑制剂
      ≥10.65 mg/mL
      insoluble in H2O
  8. Dronedarone
    A3374 Dronedarone
    中文名: 决奈达隆
    Target: Cytochrome P450 (CYP450)|sodium channel|adrenergic receptor|potassium channel|calcium channel
    Summary: CYP3A4和2D6抑制剂
      ≥27.84 mg/mL
      insoluble in H2O
  9. YM155
    A4221 YM155
     2 Citation
    Target: Survivin
    Summary: Survivin抑制剂,细胞凋亡抑制剂
      ≥22.15 mg/mL
      ≥96.2 mg/mL
  10. GDC-0449 (Vismodegib)
    A3021 GDC-0449 (Vismodegib)
     1 Citation
    中文名: 维莫德吉
    Target: P-glycoprotein (P-gp)|Hedgehog
    Summary: Hedgehog拮抗剂
      ≥21.08 mg/mL
      insoluble in H2O

10 件产品

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