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Signaling Pathways - Selective - SGLT - ROS1 - Voltage-gated Sodium (NaV) Channels

11件产品中的 1-10

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  1. Entrectinib
    B5859 Entrectinib
    中文名: 恩曲替尼
    Target: Trk Receptors|ALK|ROS1
    Summary: ALK激酶抑制剂
      ≥28.05 mg/mL
      insoluble in H2O
  2. PF-06463922
    B4882 PF-06463922
    中文名: 劳拉替尼
    Target: ALK|ROS1
    Summary: ALK/ROS1的强效选择性抑制剂
      ≥20.3 mg/mL
      insoluble in H2O
  3. ProTx II
    B5515 ProTx II
    Target: Voltage-gated Sodium (NaV) Channels
    Summary: NaV1.7通道阻断剂
      Soluble to 1 mg/mL
  4. Quinidine
    B7590 Quinidine
    中文名: 奎尼丁
    Target: Voltage-gated Sodium (NaV) Channels|Cytochrome P450 (CYP450)
    Summary: 降低Na+和K+通道电流
      ≥11.95 mg/mL
      insoluble in H2O
  5. Phenytoin sodium
    B2272 Phenytoin sodium
    中文名: 苯妥英钠
    Target: Voltage-gated Sodium (NaV) Channels
    Summary: 钠通道稳定剂
      ≥11.55 mg/mL
      insoluble in H2O
  6. Proparacaine HCl
    B2274 Proparacaine HCl
    中文名: 盐酸丙美卡因
    Target: Voltage-gated Sodium (NaV) Channels
    Summary: 电压门控钠通道拮抗剂
      ≥14.9 mg/mL
      ≥17.73 mg/mL
  7. A-803467
    B2277 A-803467
    Target: Voltage-gated Sodium (NaV) Channels
    Summary: NaV1.8通道阻断剂
      ≥13.95 mg/mL
      insoluble in H2O
  8. Canagliflozin
    A8333 Canagliflozin
     1 Citation
    中文名: 卡格列净
    Target: SGLT
    Summary: SGLT2的有效选择性抑制剂
      ≥22.25 mg/mL
      insoluble in H2O
  9. Zonisamide
    A5354 Zonisamide
    中文名: 唑尼沙胺
    Target: Voltage-gated Sodium (NaV) Channels|Voltage-gated Calcium Channels (CaV)|Carbonic Anhydrases|Calcium-Activated Potassium (KCa) Channels
    Summary: 抗惊厥和机械效应的抗癫痫药
      ≥8.35 mg/mL
      insoluble in H2O
  10. Phloretin
    A3723 Phloretin
    中文名: 根皮素
    Target: SGLT
    Summary: 在苹果中发现的二氢查耳酮
      ≥105 mg/mL
      insoluble in H2O

11件产品中的 1-10

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