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Signaling Pathways - Aldosterone receptor - Voltage-gated Sodium (NaV) Channels - PARs - Animal Experiments

10 件产品

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  1. SCH 79797 dihydrochloride
    B6801 SCH 79797 dihydrochloride
    Target: PARs
    Summary: PAR1受体拮抗剂
      Soluble in DMSO
  2. Quinidine
    B7590 Quinidine
    中文名: 奎尼丁
    Target: Voltage-gated Sodium (NaV) Channels|Cytochrome P450 (CYP450)
    Summary: 降低Na+和K+通道电流
      ≥11.95 mg/mL
      insoluble in H2O
  3. Bupivacaine HCl
    B1420 Bupivacaine HCl
    中文名: 盐酸布比卡因
    Target: Voltage-gated Sodium (NaV) Channels
    Summary: 麻醉药
      ≥10.25 mg/mL
      ≥16.23 mg/mL
  4. Phenytoin sodium
    B2272 Phenytoin sodium
    中文名: 苯妥英钠
    Target: Voltage-gated Sodium (NaV) Channels
    Summary: 钠通道稳定剂
      ≥11.55 mg/mL
      insoluble in H2O
  5. Proparacaine HCl
    B2274 Proparacaine HCl
    中文名: 盐酸丙美卡因
    Target: Voltage-gated Sodium (NaV) Channels
    Summary: 电压门控钠通道拮抗剂
      ≥14.9 mg/mL
      ≥17.73 mg/mL
  6. A-803467
    B2277 A-803467
    Target: Voltage-gated Sodium (NaV) Channels
    Summary: NaV1.8通道阻断剂
      ≥13.95 mg/mL
      insoluble in H2O
  7. Riluzole
    A8513 Riluzole
    中文名: 力鲁唑
    Target: Voltage-gated Sodium (NaV) Channels|glutamate release
    Summary: 钠通道抑制剂
      ≥23.4 mg/mL
      insoluble in H2O
  8. Potassium Canrenoate
    A8506 Potassium Canrenoate
    Target: Aldosterone receptor
    Summary: 醛固酮拮抗剂
      insoluble in DMSO
      ≥117.4 mg/mL
  9. Zonisamide
    A5354 Zonisamide
    中文名: 唑尼沙胺
    Target: Voltage-gated Sodium (NaV) Channels|Voltage-gated Calcium Channels (CaV)|Carbonic Anhydrases|Calcium-Activated Potassium (KCa) Channels
    Summary: 抗惊厥和机械效应的抗癫痫药
      ≥8.35 mg/mL
      insoluble in H2O
  10. Flecainide acetate
    A3418 Flecainide acetate
    中文名: 氟卡胺
    Target: Voltage-gated Sodium (NaV) Channels
    Summary: 抗心律失常药
      ≥47.4 mg/mL
      ≥23.7 mg/mL

10 件产品

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