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Signaling Pathways - Calpains - Voltage-gated Potassium (KV) Channels - Sir2-like Family Deacetylases (Sirtuins) - Animal Experiments

15件产品中的 1-10

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  1. Inauhzin
    B3272 Inauhzin
    Target: Sir2-like Family Deacetylases (Sirtuins)
    Summary: SIRT1抑制剂
      ≥23.5 mg/mL
      insoluble in H2O
  2. Psora 4
    B7659 Psora 4
     1 Citation
    Target: Voltage-gated Potassium (KV) Channels
    Summary: Kv1.3阻断剂
      ≥15.75 mg/mL
      insoluble in H2O
  3. Ibutilide Fumarate
    B2278 Ibutilide Fumarate
    中文名: 富马酸伊布利特
    Target: Voltage-gated Potassium (KV) Channels|Voltage-gated Calcium Channels (CaV)|sodium channel
    Summary: III类抗心律失常药物
      ≥25.6 mg/mL
      ≥16.4 mg/mL
  4. Cisapride
    B1198 Cisapride
    Target: Voltage-gated Potassium (KV) Channels|5-HT4 Receptor
    Summary: 5-HT4受体激动剂
      ≥23.3 mg/mL
      insoluble in H2O
  5. Terfenadine
    A8534 Terfenadine
    中文名: 特非那定
    Target: Voltage-gated Potassium (KV) Channels|Histamine H1 Receptors|Inward Rectifier Potassium (Kir) Channels
    Summary: 组胺H1受体拮抗剂
      ≥18 mg/mL
      insoluble in H2O
  6. Tenovin-6
    A8302 Tenovin-6
    Target: Sir2-like Family Deacetylases (Sirtuins)
    Summary: SIRT抑制剂,p53激活剂
      ≥22.75 mg/mL
      insoluble in H2O
  7. PD 150606
    A4413 PD 150606
    Target: Calpains
    Summary: 非肽类钙蛋白酶抑制剂
      Soluble in DMSO
  8. MDL 28170
    A4412 MDL 28170
    Target: Cathepsins|Calpains
    Summary: Calpain和cathepsin B抑制剂
      ≥16.75 mg/mL
      insoluble in H2O
  9. SRT2104 (GSK2245840)
    A3821 SRT2104 (GSK2245840)
     1 Citation
    Target: Sir2-like Family Deacetylases (Sirtuins)
    Summary: SIRT1激活剂
      ≥6.46 mg/mL
      insoluble in H2O
  10. Tenovin-1
    A4203 Tenovin-1
    Target: Sir2-like Family Deacetylases (Sirtuins)|p53|p21
    Summary: SIRT2 抑制剂,p53激活剂
      ≥15 mg/mL
      insoluble in H2O

15件产品中的 1-10

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